Product Name : (±)-EvodiamineDescription:(±)-Evodiamine, a quinazolinocarboline alkaloid, is a Top1 inhibitor. Evodiamine exhibits anti-inflammatory, antiobesity, and antitumor effects. (±)-Evodiamine inhibits the proliferation of a wide variety of tumor cells by…
Product Name : FLAG tag PeptideDescription:A fusion tag called FLAG and consisting of eight amino acids Asp-Tyr-Lys-Asp-Asp-Asp-Asp-Lys including an enterokinase-cleavage site, was specifically designed for immunoaffinity chromatography. It allows elution…
Product Name : InupadenantDescription:Inupadenant is an orally active, highly selective A2A receptor antagonist. Inupadenant is not brain-penetrant. Inupadenant has potent anti-tumor activity.CAS: 2246607-08-7Molecular Weight:604.65Formula: C25H26F2N8O4S2Chemical Name: 7-amino-10-ethoxy]phenyl]piperazin-1-yl]ethyl]-4-(furan-2-yl)-12-thia-3, 5, 6, 8,…
Product Name : KA2507Description:KA2507 is a potent and selective HDAC6 inhibitor, with an IC50 of 2.5 nM. KA2507 shows antitumor activities and immune modulatory effects in preclinical models.CAS: 1636894-46-6Molecular Weight:322.32Formula:…
Product Name : Methyl citrateDescription:Methyl citrate is a Monoamine oxidase B (MAO-B) inhibitor (IC50=0.23 mM). Methyl citrate is isolated from the fruits of Opuntia ficus-indica var. saboten Makino.CAS: 26163-61-1Molecular Weight:204.13Formula:…
Product Name : UC-112Description:UC-112 is an IAP inhibitor. It acts by suppressing X-linked inhibitor of apoptosis protein (XIAP) and survivin levels, inhibiting the growth of P-glycoproteins, and activating caspase-3/7 and…
Product Name : AG-014699(PF-01367338)Description:Rucaparib (AG014699) is an orally active and potent inhibitor of PARP with Ki of 1.4 nM for PARP1 in a cell-free assay. Rucaparib shows binding affinity to…
Product Name : TacrolimusDescription:Tacrolimus (FK506), a macrocyclic lactone, binds to FK506 binding protein (FKBP) to form a complex. Tacrolimus inhibits calcineurin phosphatase, which inhibits T-lymphocyte signal transduction and IL-2 transcription.…
Product Name : ASTX-029Description:ASTX-029 is an orally bioavailable inhibitor of the extracellular signal-regulated kinases (ERK) 1 and 2, with potential antineoplastic activity. ASTX-029 inhibits ERK-dependent tumor cell proliferation and survival.CAS:…
Product Name : CID-16020046Description:CID-16020046 is a selective GPR55 LPI receptor antagonist with IC50 of 015 MCAS: 834903-43-4Molecular Weight:425.44Formula: C25H19N3O4Chemical Name: 4-pyrazol-5-yl]benzoic acidSmiles : CC1C=CC(=CC=1)C1=NNC2=C1C(C1=CC(O)=CC=C1)N(C1C=CC(=CC=1)C(O)=O)C2=OInChiKey: VGUQVYZXABOXCX-UHFFFAOYSA-NInChi : InChI=1S/C25H19N3O4/c1-14-5-7-15(8-6-14)21-20-22(27-26-21)24(30)28(18-11-9-16(10-12-18)25(31)32)23(20)17-3-2-4-19(29)13-17/h2-13,23,29H,1H3,(H,26,27)(H,31,32)Purity: ≥98% (or refer…