Calcitriol D6
Product Name : Calcitriol D6Description:Calcitriol D6 is the deuterated form of Calcitriol(1,25-Dihydroxyvitamin D3; Rocaltrol ), which is the hormonally active form of vitamin D, Calcitriol is the active metabolite of…
November 2024
cis, cis-Muconic acid
Product Name : cis, cis-Muconic acidDescription:cis,cis-Muconic acid, a metabolic intermediate of Klebsiella pneumonia, can be converted to adipic acid and terephthalic acid, which are important monomers of synthetic polymers. cis,cis-Muconic…
Nav1.1 activator 1
Product Name : Nav1.1 activator 1Description:Nav1.1 activator 1 (compound 4), a highly potent Nav1.1 activator with BBB penetration, increases decay time constant (tau) of Nav1.1 currents at 0.03 μM along…
Vps34-IN-1
Product Name : Vps34-IN-1Description:Vps34-IN-1 is an inhibitor of Vps34 extracted from patent WO2012085815A1, compound example 16a, with an IC50 of 4 nM. Vps34-IN-1 modulates autophagy.CAS: 1383716-33-3Molecular Weight:425.91Formula: C21H24ClN7OChemical Name: 1-({2--4′-(cyclopropylmethyl)--2′-yl}amino)-2-methylpropan-2-olSmiles…
G-5555
Product Name : G-5555Description:G-5555 is a potent p21-activated kinase 1 (PAK1) inhibitor with Kis of 3.7 nM and 11 nM for PAK1 and PAK2, respectively.CAS: 1648863-90-4Molecular Weight:492.96Formula: C25H25ClN6O3Chemical Name: 6--2-(methylamino)-8-{methyl}-7H,8H-pyridopyrimidin-7-oneSmiles…
PHCCC
Product Name : PHCCCDescription:PHCCC is a Group I mGluR antagonist with an IC50 of 3 μM. PHCCC is a selective positive modulator of mGlu4 receptor. Antiparkinsonian effect.CAS: 179068-02-1Molecular Weight:294.30Formula: C17H14N2O3Chemical…
Raloxifene 6, 4′-Bis-β-D-glucuronide
Product Name : Raloxifene 6, 4′-Bis-β-D-glucuronideDescription:Raloxifene 6,4′-Bis-β-D-glucuronide (compound IV) is a metabolite of Raloxifene. Raloxifene is a selective estrogen receptor antagonist for the prevention of osteoporosis.CAS: 182507-20-6Molecular Weight:825.83Formula: C40H43NO16SChemical Name:…
Ipragliflozin
Product Name : IpragliflozinDescription:Ipragliflozin, also known as ASP1941, is a potent and selective SGLT2 inhibitor for treatment of type 2 diabetes. Ipragliflozin treatment improved glycaemic control when added to metformin…
BA38017
Product Name : BA38017Description:BA38017 is a potent HBV core protein assembly modulator. BA38017 inhibits HBV replication with an EC50 of 0.20 μM.CAS: 1333905-67-1Molecular Weight:307.70Formula: C15H11ClFNO3Chemical Name: Smiles : O=C(NC1=CC(Cl)=C(F)C=C1)C1=CC=CC2OCCOC=21InChiKey: JAVDMGUBEXUDIH-UHFFFAOYSA-NInChi…
Hetrombopag
Product Name : HetrombopagDescription:Hetrombopag is an orally active human thrombopoietin receptor agonist. Hetrombopag protects Cardiomyocyte Survival from Oxidative Stress Damage as an Enhancer of Stem Cells. Hetrombopag specifically stimulated proliferation…