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Year: 2024

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(±)-Evodiamine

Product Name : (±)-EvodiamineDescription:(±)-Evodiamine, a quinazolinocarboline alkaloid, is a Top1 inhibitor. Evodiamine exhibits anti-inflammatory, antiobesity, and antitumor effects. (±)-Evodiamine inhibits…

pyruvate-dehydrogenase inhibitorDecember 31, 2024
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FLAG tag Peptide

Product Name : FLAG tag PeptideDescription:A fusion tag called FLAG and consisting of eight amino acids Asp-Tyr-Lys-Asp-Asp-Asp-Asp-Lys including an enterokinase-cleavage…

pyruvate-dehydrogenase inhibitorDecember 30, 2024
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Inupadenant

Product Name : InupadenantDescription:Inupadenant is an orally active, highly selective A2A receptor antagonist. Inupadenant is not brain-penetrant. Inupadenant has potent…

pyruvate-dehydrogenase inhibitorDecember 29, 2024
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KA2507

Product Name : KA2507Description:KA2507 is a potent and selective HDAC6 inhibitor, with an IC50 of 2.5 nM. KA2507 shows antitumor…

pyruvate-dehydrogenase inhibitorDecember 28, 2024
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Methyl citrate

Product Name : Methyl citrateDescription:Methyl citrate is a Monoamine oxidase B (MAO-B) inhibitor (IC50=0.23 mM). Methyl citrate is isolated from…

pyruvate-dehydrogenase inhibitorDecember 27, 2024
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UC-112

Product Name : UC-112Description:UC-112 is an IAP inhibitor. It acts by suppressing X-linked inhibitor of apoptosis protein (XIAP) and survivin…

pyruvate-dehydrogenase inhibitorDecember 26, 2024
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AG-014699(PF-01367338)

Product Name : AG-014699(PF-01367338)Description:Rucaparib (AG014699) is an orally active and potent inhibitor of PARP with Ki of 1.4 nM for…

pyruvate-dehydrogenase inhibitorDecember 25, 2024
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Tacrolimus

Product Name : TacrolimusDescription:Tacrolimus (FK506), a macrocyclic lactone, binds to FK506 binding protein (FKBP) to form a complex. Tacrolimus inhibits…

pyruvate-dehydrogenase inhibitorDecember 24, 2024
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ASTX-029

Product Name : ASTX-029Description:ASTX-029 is an orally bioavailable inhibitor of the extracellular signal-regulated kinases (ERK) 1 and 2, with potential…

pyruvate-dehydrogenase inhibitorDecember 23, 2024
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CID-16020046

Product Name : CID-16020046Description:CID-16020046 is a selective GPR55 LPI receptor antagonist with IC50 of 015 MCAS: 834903-43-4Molecular Weight:425.44Formula: C25H19N3O4Chemical Name:…

pyruvate-dehydrogenase inhibitorDecember 22, 2024

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